Ellsworth, Edmund : rechercher sur Z-Library

Journal of Molecular Recognition

Année:

2008

Langue:

english

Fichier:

PDF, 178 KB

english, 2008

Spermine in semen of male sea lamprey acts as a sex pheromone

Scott, Anne M., Zhang, Zhe, Jia, Liang, Li, Ke, Zhang, Qinghua, Dexheimer, Thomas, Ellsworth, Edmund, Ren, Jianfeng, Chung-Davidson, Yu-Wen, Zu, Yao, Neubig, Richard R., Li, Weiming, Wolfner, Mariana

Journal:

PLoS Biology

Année:

2019

Langue:

english

Fichier:

PDF, 1.97 MB

english, 2019

Inhibitors of HIV protease: Unique non-peptide active site templates

Bradley D. Tait, John Domagala, Edmund L. Ellsworth, Donna Ferguson, Christopher Gajda, Donald Hupe, Elizabeth A. Lunney, Peter J. Tummino

Journal:

Année:

1996

Langue:

english

Fichier:

PDF, 405 KB

english, 1996

Synthesis and Structural—Activity Relationships of 3-Hydroxyquinazoline-2,4-dione Antibacterial Agents.

Tuan P. Tran, Edmund L. Ellsworth, Michael A. Stier, John M. Domagala, H. D. Hollis Showalter, Stephen J. Gracheck, Martin A. Shapiro, Themis E. Joannides, Rajeshwar Singh

Journal:

ChemInform

Année:

2004

Fichier:

PDF, 11 KB

2004

A facile synthesis of substituted 3-amino-1H-quinazoline-2,4-diones

Tuan P. Tran, Edmund L. Ellsworth, Brian M. Watson, Joseph P. Sanchez, H. D. Hollis Showalter, John R. Rubin, Michael A. Stier, Judy Yip, Dai Q. Nguyen, Paul Bird, Rajeshwar Singh

Journal:

Journal of Heterocyclic Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 124 KB

english, 2005

Discovery and optimization of nonpeptide HIV-1 protease inhibitors

Peter J. Tummino, J.V.N. Vara Prasad, Donna Ferguson, Carolyn Nouhan, Neil Graham, John M. Domagala, Edmund Ellsworth, Christopher Gajda, Susan E. Hagen, Elizabeth A. Lunney, Kimberly S. Para, Bradley

Journal:

Bioorganic & Medicinal Chemistry

Année:

1996

Langue:

english

Fichier:

PDF, 779 KB

english, 1996

Synthesis and structural–activity relationships of 3-hydroxyquinazoline-2,4-dione antibacterial agents

Tuan P. Tran, Edmund L. Ellsworth, Michael A. Stier, John M. Domagala, H.D. Hollis Showalter, Stephen J. Gracheck, Martin A. Shapiro, Themis E. Joannides, Rajeshwar Singh

Journal:

Tuan P. Tran, Edmund L. Ellsworth, Joseph P. Sanchez, Brian M. Watson, Michael A. Stier, H.D. Hollis Showalter, John M. Domagala, Martin A. Shapiro, E. Themis Joannides, Stephen J. Gracheck, Dai Q. Ng

Année:

2004

Langue:

english

Fichier:

PDF, 267 KB

english, 2004

Structure–activity relationships of 3-aminoquinazolinediones, a new class of bacterial type-2 topoisomerase (DNA gyrase and topo IV) inhibitors

Journal:

Année:

2007

Langue:

english

Fichier:

PDF, 197 KB

english, 2007

The synthesis and biological evaluation of novel series of nitrile-containing fluoroquinolones as antibacterial agents

Sean T. Murphy, Heather L. Case, Edmund Ellsworth, Susan Hagen, Michael Huband, Themis Joannides, Chris Limberakis, Keith R. Marotti, Amy M. Ottolini, Mark Rauckhorst, Jeremy Starr, Michael Stier, Cla

Journal:

Année:

2007

Langue:

english

Fichier:

PDF, 163 KB

english, 2007

Synthesis and antibacterial activity of the C-7 side chain of 3-aminoquinazolinediones

Kim M. Hutchings, Tuan P. Tran, Edmund L. Ellsworth, Brian M. Watson, Joseph P. Sanchez, H.D. Hollis Showalter, Michael A. Stier, Martin Shapiro, E. Themis Joannides, Michael Huband, Dai Q. Nguyen, Sa

Journal:

Bruce H. Lipshutz, Edmund L. Ellsworth, Teruna J. Siahaan, Ata Shirazi

Année:

2008

Langue:

english

Fichier:

PDF, 174 KB

english, 2008

Unexpected affects of Me3Si-X on reactions of higher order cyanocuprates

Journal:

Bruce H. Lipshutz, Edmund L. Ellsworth, James R. Behling, Arthur L. Campbell

Année:

1988

Langue:

english

Fichier:

PDF, 256 KB

english, 1988

Effects of gengenions on organocuprate reactivity/selectivity: Higher order, mixed lithio-sodio cyanocuprates

Journal:

Bruce H. Lipshutz, Edmund L. Ellsworth, Stuart H. Dimock, Deborah C. Reuter

Année:

1988

Langue:

english

Fichier:

PDF, 242 KB

english, 1988

Transmetalation reactions of higher order cyanocuprates: Direct formation of trialkyltin cuprates from tin hydrides which bypasses organolithium intermediates

Journal:

Année:

1989

Langue:

english

Fichier:

PDF, 206 KB

english, 1989

Nonpeptidic HIV protease inhibitors: 6-alkyl-5, 6-dihydropyran-2-ones possessing achiral 3-(4-amino/carboxamide-2-t-butyl, 5-methylphenyl thio) moiety: Antiviral activities and pharmacokinetic properties

J.V.N. Vara Prasad, Fred E. Boyer, John M. Domagala, Edmund L. Ellsworth, Christopher Gajda, Susan E. Hagen, Larry J. Markoski, Bradley D. Tait, Elizabeth A. Lunney, Peter J. Tummino, Donna Ferguson,

Journal:

Année:

1999

Langue:

english

Fichier:

PDF, 335 KB

english, 1999

4-Hydroxy-5,6-Dihydro-2H-pyran-2-ones. 3. Bicyclic and hetero-aromatic ring systems as 3-position scaffolds to bind to S1′ and S2′ of the HIV-1 protease enzyme

Edmund L. Ellsworth, John Domagala, J.V.N. Vara Prasad, Susan Hagen, Donna Ferguson, Tod Holler, Donald Hupe, Neil Graham, Caroline Nouhan, Peter J. Tummino, Greg Zeikus, Elizabeth A. Lunney

Journal:

Année:

1999

Langue:

english

Fichier:

PDF, 342 KB

english, 1999

Nonpeptidic HIV protease inhibitors: 6-alkyl-5,6-dihydropyran-2-ones possessing a novel and achiral 3-(2-t-butyl-5-methyl-4-sulfamate)phenylthio moiety

J.V.N Vara Prasad, Larry J Markoski, Fred E Boyer, John M Domagala, Edmund L Ellsworth, Christopher Gajda, Susan E Hagen, Bradley D Tait, Elizabeth A Lunney, Peter J Tummino, Donna Ferguson, Tod Holle

Journal:

J.V.N. Vara Prasad, Frederick E. Boyer, John M. Domagala, Edmund L. Ellsworth, Christopher Gajda, Harriet W. Hamilton, Susan E. Hagen, Larry J. Markoski, Bruce A. Steinbaugh, Bradley D. Tait, Christin

Année:

1999

Langue:

english

Fichier:

PDF, 336 KB

english, 1999

Nonpeptidic HIV protease inhibitors possessing excellent antiviral activities and therapeutic indices. PD 178390: a lead HIV protease inhibitor

Journal:

Bioorganic & Medicinal Chemistry

Année:

1999

Langue:

english

Fichier:

PDF, 468 KB

english, 1999

Nonpeptidic HIV protease inhibitors: 3-(S-benzyl substituted)-4-hydroxy-6-(phenyl substituted)-2H-pyran-2-one with an inverse mode of binding

J.V.N. Vara Prasad, A. Pavlovsky, Kimberly S. Para, Edmund L. Ellsworth, Peter J. Tummino, Carolyn Nouhan, Donna Ferguson

Journal:

Année:

1996

Langue:

english

Fichier:

PDF, 331 KB

english, 1996

Synthesis of the novel antibacterial 6,8-dihydroxy-7-propyl-9H-pyrrolo[1,2-b][1,3]-benzoxazin-9-one

Liren Huang, Edmund L Ellsworth, Sab Randhawa, Michael A Stier, Yanting Huang, Paul Bird, Mikhail Lebedev, Kun Wu, Ron G Micetich, John M Domagala, Rajeshwar Singh, Norm L Colbry

Journal:

Edmund L. Ellsworth, et al. et al.

Année:

2000

Langue:

english

Fichier:

PDF, 134 KB

english, 2000

ChemInform Abstract: Synthesis of the Novel Antibacterial 6,8-Dihydroxy-7-propyl-9H-pyrrolo[1,2-b][1,3]-benzoxazin-9-one.

Journal:

ChemInform

Année:

2000

Fichier:

PDF, 28 KB

2000

Stereoselective Synthesis of ( S )-3-(Methylamino)-3-(( R )-pyrrolidin-3-yl)propanenitrile

Lall, Manjinder S., Hoge, Garrett, Tran, Tuan P., Kissel, William, Murphy, Sean T., Taylor, Clarke, Hutchings, Kim, Samas, Brian, Ellsworth, Edmund L., Curran, Timothy, Showalter, H. D. Hollis

Journal:

Journal of Organic Chemistry

Année:

2012

Langue:

english

Fichier:

PDF, 445 KB

english, 2012

3-Aminoquinazolinediones as a New Class of Antibacterial Agents Demonstrating Excellent Antibacterial Activity Against Wild-Type and Multidrug Resistant Organisms

Ellsworth, Edmund L., Tran, Tuan P., Hollis Showalter, H. D., Sanchez, Joseph P., Watson, Brian M., Stier, Michael A., Domagala, John M., Gracheck, Stephen J., Joannides, E. Themis, Shapiro, Martin A.

Journal:

Lipshutz, Bruce H., Ellsworth, Edmund L., Dimock, Stuart H.

Année:

2006

Langue:

english

Fichier:

PDF, 48 KB

english, 2006

On the composition of Yamamoto's reagent: "RCu.cntdot.BF3"

Journal:

Lipshutz, Bruce H., Sharma, Sunaina, Ellsworth, Edmund L.

Année:

1990

Langue:

english

Fichier:

PDF, 413 KB

english, 1990

Higher order cyanocuprates R2Cu(CN)Li2: discrete reagents or lower order lithium cyanide (LiCN) modified Gilman cuprates?

Journal:

Edmund Otis Hovey, A. P. Brigham, Isaiah Bowman, George C. Curtis, W. M. Davis, N. M. Fenneman, Ellsworth Huntington, William Libbey, Lawrence Martin, Ralph S. Tarr, Cleveland Abbe, Alfred H. Brooks,

Année:

1990

Langue:

english

Fichier:

PDF, 427 KB

english, 1990

Second Annual Meeting of the Association of American Geographers: Papers and Abstracts

Journal:

Bulletin of the American Geographical Society

Année:

1906

Langue:

english

Fichier:

PDF, 1.39 MB

english, 1906

5,6-Dihydropyran-2-ones Possessing Various Sulfonyl Functionalities: Potent Nonpeptidic Inhibitors of HIV Protease

Boyer, Frederick E., Vara Prasad, J. V. N., Domagala, John M., Ellsworth, Edmund L., Gajda, Christopher, Hagen, Susan E., Markoski, Larry J., Tait, Bradley D., Lunney, Elizabeth A., Palovsky, Alexande

Journal:

Lipshutz, Bruce H., Ellsworth, Edmund L., Dimock, Stuart H., Smith, Robin A. J.

Année:

2000

Langue:

english

Fichier:

PDF, 428 KB

english, 2000

New methodology for conjugate additions of allylic ligands to .alpha.,.beta.-unsaturated ketones: synthetic and spectroscopic studies

Journal:

Année:

1990

Langue:

english

Fichier:

PDF, 1.04 MB

english, 1990

4-Hydroxy-5,6-dihydropyrones. 2. Potent Non-Peptide Inhibitors of HIV Protease

Tait, Bradley D., Hagen, Susan, Domagala, John, Ellsworth, Edmund L., Gajda, Christopher, Hamilton, Harriet W., Vara Prasad, J. V. N., Ferguson, Donna, Graham, Neil, Hupe, Donald, Nouhan, Carolyn, Tum

Journal:

Lipshutz, Bruce H., Ellsworth, Edmund L., Dimock, Stuart H., Smith, Robin A. J.

Année:

1997

Langue:

english

Fichier:

PDF, 330 KB

english, 1997

Understanding allylic organocuprates: .sigma.- or .pi.-bound reagents?

Journal:

Journal of Organic Chemistry

Année:

1989

Langue:

english

Fichier:

PDF, 826 KB

english, 1989

Fine tuning the silicon-tin bond: transmetalations forming either trialkylstannyl or trialkylsilyl higher order cyanocuprates

Lipshutz, Bruce H., Reuter, Deborah C., Ellsworth, Edmund L.

Journal:

Journal of Organic Chemistry

Année:

1989

Langue:

english

Fichier:

PDF, 329 KB

english, 1989

The discovery of isoxazoline oxime ethers as a new class of ectoparasiticides for the control of Haematobia irritans (horn fly) in cattle

Curtis, Michael P., Chubb, Nathan, Ellsworth, Edmund, Goodwin, Richard, Holzmer, Sue, Koch, Jason, McTier, Tom, Menon, Sanjay, Mills, Kent, Pullins, Aleah, Stuk, Tim, Zinser, Erich

Journal:

Lipshutz, Bruce H., Ellsworth, Edmund L., Siahaan, Teruna J.

Année:

2014

Langue:

english

Fichier:

PDF, 1.19 MB

english, 2014

Effects of boron trifluoride etherate on higher order organocuprate reactions: substrate activation or cuprate modification?

Journal:

Hagen, Susan E., Vara Prasad, J. V. N., Boyer, Frederick E., Domagala, John M., Ellsworth, Edmund L., Gajda, Christopher, Hamilton, Harriet W., Markoski, Larry J., Steinbaugh, Bruce A., Tait, Bradley

Année:

1988

Langue:

english

Fichier:

PDF, 269 KB

english, 1988

Synthesis of 5,6-Dihydro-4-hydroxy-2- pyrones as HIV-1 Protease Inhibitors: The Profound Effect of Polarity on Antiviral Activity

Journal:

Lipshutz, Bruce H., Ellsworth, Edmund L.

Année:

1997

Langue:

english

Fichier:

PDF, 157 KB

english, 1997

Hydrozirconation-transmetalation. A mild, direct route to higher order vinylic cuprates from monosubstituted acetylenes

Journal:

Lipshutz, Bruce H., Crow, Robert, Dimock, Stuart H., Ellsworth, Edmund L., Smith, Robin A. J., Behling, James R.

Année:

1990

Langue:

english

Fichier:

PDF, 276 KB

english, 1990

Ligand exchange between cyanocuprates and allylic stannanes: a novel, direct route to allylic cuprates possessing remarkable reactivity and stability

Journal: